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Search Results for " water solubility "

25

阻害剤

5

天然化合物

3

リコンビナントタンパク質

カタログ番号 製品名 別名 ターゲット
T24493 Monoelaidin
Monoelaidin is a poorly water-soluble drug enhancer of solubility and oral bioavailability.
T4545 Propacetamol Hydrochloride Propacetamol HCL Others
Propacetamol Hydrochloride (Propacetamol HCL) is a prodrug of paracetamol (acetaminophen) with improved water solubility. Propacetamol Hydrochloride is an analgesic drug delivered by IV when the oral application of NSAID...
T50013 4-[(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]benzoic acid Others
4-[(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]benzoic acid is a synthetic compound with potent antitumor activity, high efficiency and selectivity against tumor cells. However, it has poor solubility in water and is pot...
T14589 Biotin-PEG3-acid Others , PROTAC Linker
Biotin-PEG3-acid is a biotin-labeled, PEG-based PROTAC linker that can be used in the synthesis of PROTACs.Biotin-PEG3-acid is a heterobiofunctional biotin PEG derivative containing a carboxylic acid group. The hydrophil...
T14050 5-FAM 5-Carboxyfluorescein Others
5-FAM (5-Carboxyfluorescein) (5-Carboxyfluorescein) contains a carboxylic acid, which can be used to react with primary amines via carbodiimide activation of the carboxylic acid. Fluorescein is the most common fluorescen...
T33606 NBI-30545
NBI-30545 is a potent corticotropin-releasing factor-1 antagonist with sufficient lipophilicity and water solubility for the treatment of stress disorders.
T6538 Hydroxypropyl Cellulose Others
Hydroxypropyl cellulose (HPC) is a derivative of cellulose with both water solubility and organic solubility, it is used as food additive and sieving matrix for DNA separations.
T19167 8pyDTZ Others
T80936 Trisulfo-Cy3-acid disodium
Trisulfo-Cy3-acid disodium, a Cy3 (Cyanine3) dye derivative, possesses three sulfonate ions and exhibits enhanced water solubility.
T69608 TG11-77 HCl
TG11-77 HCl is a novel, Potent, Selective, Water Soluble, Brain-Permeable EP2 Receptor Antagonist. TG11-77 HCl has a Schild KB of 9.7 nM on EP2, a water solubility of 2.5 mM, a brain-to-plasma ratio of 0.4, and a plasma...
T81067 Sulfo-Cy3(Me)COOH sodium
Sulfo-Cy3(Me)COOH sodium and Trisulfo-Cy3-acid disodium are sulfonated derivatives of the Cyanine3 (Cy3) dye; the introduction of sulfonate ions enhances their water solubility.
T69609 TG11-77 free base
TG11-77 free base is a novel, Potent, Selective, Water Soluble, Brain-Permeable EP2 Receptor Antagonist. TG11-77 free base has a Schild KB of 9.7 nM on EP2, a water solubility of 2.5 mM, a brain-to-plasma ratio of 0.4, ...
T30538 BMS-695735 CHEMBL459729,DNC008930,BMS 695735,BMS695735,BDBM27888
BMS-695735, a benzimidazole inhibitor of insulin-like growth factor-1 receptor, has broad-spectrum antitumor activity in vivo. It was found that BMS-695735 had strong inhibition of CYP3A4, induction of CYP3A4 mediated by...
T82852 BMI-Glu
BMI-Glu, a selective γ-glutamyl transpeptidase (GGT) fluorescent probe, exhibits a Michaelis constant (Km) of 69.63 µM and is characterized by its high sensitivity, good water solubility, and biocompatibility [1].
T18940 Cy2 CY2 Non-Sulfonated,Cyanine2 Others
Cy2 (CY2 Non-Sulfonated) is a cyanine dye with long wavelength, tunable absorption and emission, high extinction coefficient and good water solubility. Cy2 can be used to label amino groups in oligonucleotides, peptides,...
T63319 Antitubercular agent-32
Antitubercular agent-32 is a Benzothiazinone derivative that inhibits Mycobacterium tuberculosis and exhibits good metabolic stability and water solubility. Antitubercular agent-32 can act on decaprenylphosphoryl-β-D-rib...
T82866 Biotin-PEG-Biotin (MW 20000)
Biotin-PEG-Biotin (MW 20000) is a bifunctional PEG derivative featuring biotin labels at each terminal end. As an enzyme co-factor, biotin facilitates protein labeling, while PEG, known for its hydrophilic nature and low...
T71577 KOS-1584
KOS-1584 is a second-generation epothilone with potential antineoplastic activity. Epothilone KOS-1584 binds to tubulin and induces microtubule polymerization and stabilizes microtubules against depolymerization, which m...
T67948 OY-101
OY-101, an orally active compound, serves as a potent and specific inhibitor of P-glycoprotein (P-gp). It has the capability to sensitize drug-resistant tumors and counteract tumor multidrug resistance efficiently. Compa...
T68860 Iso-Fludelone
Iso-Fludelone is the third-generation epothilone B analogue with potential anti-mitotic and antineoplastic activites. Iso-fludelone binds to tubulin and induces microtubule polymerization and stabilizes microtubules agai...
T82868 Biotin-PEG-azide (MW 2000)
Biotin-PEG-azide (MW 2000) is a biotinylated polyethylene glycol (PEG) compound featuring an azide group. Biotin serves as an enzyme cofactor suitable for protein labeling. PEG, noted for its hydrophilicity and water sol...
T31657 Epothilone F
Epothilone F is a derivative or analogue of Epothilone D. Epothilone F is also an active metabolite of Epothilone D. In molecule of Epothilone F, a hydroxymethyl group is on the thiazole ring. Like taxanes, Epothilone F ...
T75337 Cy5.5-SE (DIPEA)
Cy5.5-SE (Cyanine5.5 NHS ester) DIPEA, a cyanine (CY) dye, comprises two nitrogen atoms linked by an odd number of methyl units. Characterized by long wavelength, tunable absorption and emission, high extinction coeffici...
T74120 Cy5 maleimide
Cy5 maleimide, a CY dye where CY represents Cyanine, comprises two nitrogen atoms linked by an odd number of methyl groups. Characteristics of Cyanine compounds include long wavelength, tunable absorption and emission, h...
T36400 Para-amino-Blebbistatin
para-amino-Blebbistatin is a more water-soluble form of (S)-4'-nitro-blebbistatin , which is a more stable and less phototoxic form of (-)-blebbistatin .1,2,3 (-)-Blebbistatin is a selective cell-permeable inhibitor of n...
カタログ番号 製品名 別名 ターゲット
T20597 Alginic acid Protanal LF,Snow acid algin G,Kelacid,Sazzio,Norgine Apoptosis , Autophagy , Histamine Receptor
Alginic acid (Snow acid algin G) is a natural polysaccharide extracted from brown seaweeds with anti-anaphylactic and anti-inflammatory activities. Alginic acid inhibits histamine release and can be used in the food indu...
T5749 10-Deacetyl-7-xylosyl paclitaxel 10-Deacetyl-7-xylosyltaxol,10-Deacetyltaxol 7-Xyloside,7-Xylosyl-10-deacetyltaxol,10-Deacetylpaclitaxel 7-Xyloside Others , Microtubule Associated
10-Deacetyl-7-xylosyl paclitaxel (7-Xylosyl-10-deacetyltaxol) is a Paclitaxel derivative with improved pharmacological features and higher water solubility,used in Chinese clinics to treat cancer.
T82148 Hydrogenated soya phosphatidylcholines
Hydrogenated soya phosphatidylcholines, a natural compound, enhances the controlled release of water-soluble drugs in oral drug delivery systems by improving drug loading and solubility [1].
T81026 Tectorigenin sodium sulfonate
Tectorigenin sodium sulfonate, a derivative of tectorigenin, is synthesized through sulfonation with sulfuric acid followed by neutralization in saturated saline. This compound exhibits excellent water solubility and pot...
T78465 H-γ-Glu-Gln-OH γ-Glutamylglutamine,γ-Glu-Gln
H-γ-Glu-Gln-OH, a hydrophilic peptide, serves as a drug carrier with high water solubility, robust drug-loading capacity, excellent biocompatibility, and minimal toxicity. This compound enhances tumor targeting and exhib...

Recombinant Proteins

カタログ番号 製品名 Species Expression System
TMPH-02916 SULT1A1 Protein, Mouse, Recombinant (His & Myc) Mouse E. coli
Sulfotransferase that utilizes 3'-phospho-5'-adenylyl sulfate (PAPS) as sulfonate donor to catalyze the sulfate conjugation of a wide variety of acceptor molecules bearing a hydroxyl or an amine groupe. Sulfonation incre...
TMPY-01617 SULT1B1 Protein, Human, Recombinant (His) Human E. coli
Sulfotransferase family cytosolic 1B member 1, also known as Sulfotransferase 1B1, Sulfotransferase 1B2, Thyroid hormone sulfotransferase, SULT1B1 and ST1B2, is a cytoplasm protein that belongs to the sulfotransferase 1 ...
TMPY-01616 SULT2B1 Protein, Human, Recombinant (His) Human E. coli
Sulfotransferase family cytosolic 2B member 1, also known as Sulfotransferase 2B1, ST2B1, Alcohol sulfotransferase, Hydroxysteroid sulfotransferase 2, SULT2B1 and HSST2, is a cytoplasm protein that belongs to the sulfotr...